Single doses of up to at least 32-fold (800 mg), as well as continuous therapy with 24-fold (600 mg) the usual daily dose are well tolerated. No life-threatening overdosing is known in humans, but only in animal studies with 2000- to 4000-fold doses (adjusted to body surface area).
Exemestane
Anastrozole
Salvestrol
Hexestrol
Fosfestrol
Norendoxifen
Tamoxifen
Formestane