2-Oxoquazepam, a major active<unk>  metabolite.<unk>  has an absorption half-life of 0.4 hours with a peak in plasma levels after 1.75 hours. It is eliminated both renally and through feces. The active metabolites of<unk>  are 2-oxoquazepam and N-desalkyl-2-oxoquazepam. The N-desalkyl-2-oxoquazepam metabolite has only limited pharmacological activity compared to the parent compound<unk>  and the active metabolite 2-oxoquazepam.<unk>  and its major active metabolite 2-oxoquazepam both show high selectivity for the type1 GABAA receptors. The elimination half-life range of<unk>  is between 27 and 41 hours.
Quazepam
Halazepam
Oxazepam
Triazolam
Gidazepam
Nordazepam
Bromazepam
Cinolazepam